Index/GhrelinGut Health

GHRELIN

Growth Hormone Secretagogue (endogenous) · Hunger Hormone

The hunger hormone — appetite, GH release, and gut motility.

FDA

Research Only

WADA

Banned

HALF-LIFE

~30 minutes

ROUTE

SubQ injection

SCHEDULE

Pre-meal or pre-workout

In Plain English

The hunger hormone — appetite, GH release, and gut motility.

Status & Legality

NATTY?

Not Natty

WADA banned substance. Tested athletes will fail.

FDA

Research Only

For research purposes only. Not FDA approved.

WADA

Banned

On WADA prohibited list. Use disqualifies in tested sports.

COMPOUNDING

Not from pharmacies

Not available from licensed compounding pharmacies.

PRESCRIBED

Not prescribed

Not prescribed in conventional medicine.

ROUTE

SubQ injection

Administration via subq injection.

Who It's For

GH stimulation

Appetite enhancement

Gut motility

Gastroparesis

How It Works

Ghrelin is the endogenous peptide produced by the stomach that signals hunger to the hypothalamus and stimulates GH release via the ghrelin receptor. Its gut motility effects make it relevant in gastroparesis treatment. GHRP-6 mimics ghrelin's effects on both GH and appetite. Exogenous ghrelin research focuses on cachexia and GI motility disorders.

Side Effects

01

Hunger/appetite stimulation

02

GI distress

03

Cortisol elevation

04

Water retention

Common Mistakes

Using native ghrelin when GHRP-6 is more practical — GHRP-6 mimics ghrelin's effects with far better stability and predictability

Not planning around the intense hunger spike — ghrelin and ghrelin mimetics cause significant appetite stimulation; have food prepared

Expecting significant GH release without combining with a GHRH — ghrelin/GHRP provides the pulse, but GHRH amplifies it 2–5×

Drug & Supplement Interactions

GLP-1 agonists (semaglutide) — directly antagonistic on appetite signals; do not combine when weight management is the goal

Insulin — ghrelin has anti-insulin effects; monitor glucose during combined use

GH secretagogues — ghrelin is the endogenous GH-releasing signal; combining with synthetic analogs is generally synergistic

The PepVault Take

Exogenous ghrelin has a very short half-life that makes it impractical for most research applications. GHRP-6 provides the same receptor activation with better stability and is far more commonly used. Native ghrelin's most interesting application is gastroparesis — gut motility restoration — where 3× daily pre-meal injections have direct research support.

Frequently Asked Questions

Stats

ONSET50
DOCUMENTATION18
SIDE INTENSITY49
CYCLE EASE70
POPULARITY25
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Sources & Studies

1/2
Real human support, no ticket queue.
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Research Use OnlyNot Medical AdviceNot FDA Evaluated18+ OnlyWADA Status Tracked

PepVault provides educational and research reference information only. Nothing on this site constitutes medical advice, diagnosis, or treatment. Content has not been evaluated by the U.S. Food and Drug Administration. No compound listed on this site is intended to diagnose, treat, cure, or prevent any disease or medical condition. The legality of peptide compounds varies by jurisdiction — you are solely responsible for compliance with the laws of your country or region. Certain compounds listed are prohibited under the World Anti-Doping Agency (WADA) Prohibited List; athletes subject to anti-doping regulations should independently verify status before use. This site is intended for adults 18 years of age or older. Always consult a licensed healthcare provider before using any compound.

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